Cart
sales@molnova.com
Home - Products - GPCR/G Protein - Cannabinoid Receptor - CB1R antagonist 1

CB1R antagonist 1

CAS No. 334668-69-8

CB1R antagonist 1( —— )

Catalog No. M35611 CAS No. 334668-69-8

CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 65 Get Quote
10MG 112 Get Quote
25MG 182 Get Quote
50MG 270 Get Quote
100MG 394 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    CB1R antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.
  • Description
    CB1R Allosteric modulator 5, a selective cannabinoid-1 receptor (CB1R) inverse agonist with an IC50 value of 4.2 μM and EC50 value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity.
  • In Vitro
    CB1R Allosteric modulator 5 has cannabinoid-1 receptor (CB1R) activity with an IC50value of 4.2 μM and EC50 value of ＞10 μM.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    Cannabinoid Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    334668-69-8
  • Formula Weight
    404.45
  • Molecular Formula
    C18H23F3N2O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (247.25 mM; Ultrasonic )
  • SMILES
    S(=O)(=O)(C1=CC(C(F)(F)F)=CC=C1)N2CCN(C(=O)C3CCCCC3)CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Petr Vachal, et al. 1-Sulfonyl-4-acylpiperazines as selective cannabinoid-1 receptor (CB1R) inverse agonists for the treatment of obesity. J Med Chem. 2009 Apr 23;52(8):2550-8?
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • SCH-336

    SCH-336 is a CB2 receptor agonist (Ki-1.8 nM, EC50-2 nM) with effective, selective, and oral activity. SCH-336 is also bioactive against CB1 receptor, and is 100 times more selective to CB2 receptor than CB1.

  • TM38837

    TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.

  • Cardiogenol C hydroc...

    Cardiogenol C hydrochloride is a cardiomyogenesis inducer in embryonic stem cells.

Sign In Join Free